LP 922761_1454808-95-7_L473433_【莱耀标准品网】

产品基本信息

产品编号：L473433

产品名称：LP 922761

产品CAS：1454808-95-7

规格含量：2.5mg

产品价格：面议

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产品详细介绍

标准品编号:	L473433
名称:	LP 922761
别名:	tert-Butyl(2-((3-(4-carbamoylphenyl)imidazo[1,2-b]pyridazin-6-yl)amino)ethyl)(methyl)carbamate
CAS号:	1454808-95-7
分子式:	C₂₁H₂₆N₆O₃
分子量:	410.47
种类:	Standards; Enzyme Activators and Inhibitors;
应用:	LP 922761 is a potent AAK1 inhibitor (IC50 values are 4.8 and 7.6 nM in enzyme and cell assays, respectively). Exhibits some selectivity for AAK1 over BIKE, and exhibits no significant activity at opioid, adrenergic α2 or GABAA receptors. Orally bioavailable. Peripherally restricted.
参考文献	Lanthorn, Thomas Herbert., et al.: PCT Int. Appl.(2013),WO2013134336A220130912.

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