产品编号:A112580
产品规格:10mg
产品价格:面议
| 标准品编号: | A112580 |
| 名称: | ABT 888 |
| 别名: | 2-[(2R)-2-Methyl-2-pyrrolidinyl]-1H-benzimidazole-7-carboxamide; A 861695; |
| CAS号: | 912444-00-9 |
| 分子式: | C₁₃H₁₆N₄O |
| 状态: | 白色至Dark Yellow Solid |
| 熔点: | >173°C (dec.) |
| 分子量: | 244.29 |
| 储存: | 冰箱保存 |
| 溶解性: | Methanol (Slightly, Heated), THF (Slightly, Heated) |
| 类别: | Research Tools; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites; |
| 应用: | ABT-888 is a potent, orally bioavailable PARP-1/-2 inhibitor shown to potentiate DNA damaging agents. The ability to potentiate temozolomide (TMZ) and develop a biological marker for PARP inhibition was evaluated in vivo. Potent PARP inhibitor. |
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