产品编号：C781420

产品规格：10mg

产品价格：面议

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产品详情

标准品编号:	C781420
名称:	CP 945598 Hydrochloride
别名:	1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)-4-piperidinecarboxamide Hydrochloride; 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)-4-piperidinecarboxamide Monohydrochloride; CP 945598; CP 945598-01; Otenabant Hydrochloride;
CAS号:	686347-12-6
参考CAS:	686344-29-6-free base
分子式:	C₂₅H₂₆Cl₃N₇O
外观:	白色固体
熔点:	283-291°C
分子量:	546.88
储存:	冰箱保存
溶解度:	DMSO (Sparingly), Methanol (Sparingly)
类别:	Standards; Controlled Substances and Drugs of Abuse for Forensic Testing;
应用:	CP 945598 is a selective, high affinity CB1 antagonist (Ki values are 0.7 and 0.12 nM in binding and functional assays respectively). Displays low affinity for CB2 receptors (Ki = 7600 nM).
参考文献	Griffith, et al.: J. Med. Chem., 52, 234 (2009), Hadcock, et al.: Biochem. Biophys. Res. Commun., 394, 366 (2010),