产品编号:D456460
产品规格:5mg
产品价格:面议
| 标准品编号: | D456460 |
| 名称: | 5-(3,5-Dimethyl-4-isoxazolyl)-1-[2-(4-morpholinyl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-benzimidazole Hydrochloride |
| 别名: | PF-CBP1; PF-06670910 |
| CAS号: | 2070014-93-4 |
| 参考CAS号: | Free Base: 1962928-21-7 |
| 分子式: | C₂₉H₃₇ClN₄O₃ |
| 分子量: | 525.08 |
| 种类: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | 5-(3,5-Dimethyl-4-isoxazolyl)-1-[2-(4-morpholinyl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-benzimidazole Hydrochloride is a potent and selective bromodomain of CREB binding protein (CBP BRD) inhibitor. 5-(3,5-Dimethyl-4-isoxazolyl)-1-[2-(4-morpholinyl)ethyl]-2-[2-(4-propoxyphenyl)ethyl]-1H-benzimidazole Hydrochloride downregulates inflammatory genes in macrophages and has therapeutic potential for treating neurological disorders. |
| 参考文献 | |