产品编号:K145558
产品规格:5mg
产品价格:面议
| 标准品编号: | K145558 |
| 名称: | KCC 07 |
| 别名: | 3-[[4-(2-Pyridinyl)-2-thiazolyl]amino]phenol |
| CAS号: | 315702-75-1 |
| 分子式: | C₁₄H₁₁N₃OS |
| 分子量: | 269.32 |
| 种类: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | KCC 07 is a MBD2 (Methyl-CpG-binding domain protein 2) inhibitor. Prevents binding of MBD2 to methylated DNA and activates brain specific angiogenesis inhibitor 1 (BAI1)/p53 signaling. Inhibits medulloblastoma (MB) cell growth in vitro and reduces tumor size in mice bearing MB xenografts. Brain penetrant. |
| 参考文献 | |