产品编号：L473433
产品规格：2.5mg
产品价格：面议
| 标准品编号: | L473433 |
| 名称: | LP 922761 |
| 别名: | tert-Butyl(2-((3-(4-carbamoylphenyl)imidazo[1,2-b]pyridazin-6-yl)amino)ethyl)(methyl)carbamate |
| CAS号: | 1454808-95-7 |
| 分子式: | C₂₁H₂₆N₆O₃ |
| 分子量: | 410.47 |
| 种类: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | LP 922761 is a potent AAK1 inhibitor (IC50 values are 4.8 and 7.6 nM in enzyme and cell assays, respectively). Exhibits some selectivity for AAK1 over BIKE, and exhibits no significant activity at opioid, adrenergic α2 or GABAA receptors. Orally bioavailable. Peripherally restricted. |
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