产品编号:M199800
产品规格:10mg
产品价格:面议
| 标准品编号: | M199800 |
| 名称: | MDV 3100 (Enzalutamide) |
| 别名: | 4-[3-[4-Cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-N-methylbenzamide; MDV3100; MDV-3100; Enzalutamide; |
| CAS号: | 915087-33-1 |
| 分子式: | C₂₁H₁₆F₄N₄O₂S |
| 外观: | 白色至白色固体 |
| 熔点: | 198 - 200°C |
| 分子量: | 464.44 |
| 储存: | 冰箱 |
| 溶解度: | Chloroform (Slightly), DMSO (Slightly), Methanol (Slightly, Heated) |
| 种类: | Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites; |
| 应用: | MDV 3100 is an androgen-receptor antagonist that blocks androgens from binding to the androgen receptor and prevents nuclear translocation and co-activator recruitment of the ligand-receptor complex. MDV 3100 has also been shown to induce tumor cell apoptosis, and has no agonist activity. MDV 3100 is a candidate for the treatment of castration-resistant prostate cancer. |
| 参考文献 | |