MDV 3100 (Enzalutamide)

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产品编号:M199800

产品规格:10mg

产品价格:面议


产品详情

标准品编号: M199800
名称: MDV 3100 (Enzalutamide)
别名: 4-[3-[4-Cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-N-methylbenzamide; MDV3100; MDV-3100; Enzalutamide;
CAS号: 915087-33-1
分子式: C₂₁H₁₆F₄N₄O₂S
外观: 白色至白色固体
熔点: 198 - 200°C
分子量: 464.44
储存: 冰箱
溶解度: Chloroform (Slightly), DMSO (Slightly), Methanol (Slightly, Heated)
种类: Standards; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites;
应用: MDV 3100 is an androgen-receptor antagonist that blocks androgens from binding to the androgen receptor and prevents nuclear translocation and co-activator recruitment of the ligand-receptor complex. MDV 3100 has also been shown to induce tumor cell apoptosis, and has no agonist activity. MDV 3100 is a candidate for the treatment of castration-resistant prostate cancer.
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