产品编号:S282318
产品规格:2.5mg
产品价格:面议
| 标准品编号: | S282318 |
| 名称: | SGC GAK 1 |
| 别名: | 6-bromo-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine |
| CAS号: | 2226517-76-4 |
| 分子式: | C₁₈H₁₇BrN₂O₃ |
| 分子量: | 389.24 |
| 类别: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | SGC GAK 1 is a high affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibited >30-fold selectivity for GAK versus a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM). |
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