XY 018

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产品编号:X746503

产品规格:2.5mg

产品价格:面议


产品详情

标准品编号: X746503
名称: XY 018
别名: N-(2'-Fluoro-4'-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-[1,1'-biphenyl]-4-yl)-2-(2-nitrophenyl)acetamide
CAS号: 1873358-87-2
分子式: C₂₃H₁₅F₇N₂O₄
分子量: 516.37
类别: Standards; Enzyme Activators and Inhibitors;
应用: XY 018 is a RORγ antagonist (EC50 = 190 nM). XY 018 suppresses androgen receptor expression in prostate cancer cell lines. Also inhibits growth of tumors in androgen receptor-positive xenograft models.
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