产品编号:X746503
产品规格:2.5mg
产品价格:面议
| 标准品编号: | X746503 |
| 名称: | XY 018 |
| 别名: | N-(2'-Fluoro-4'-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-[1,1'-biphenyl]-4-yl)-2-(2-nitrophenyl)acetamide |
| CAS号: | 1873358-87-2 |
| 分子式: | C₂₃H₁₅F₇N₂O₄ |
| 分子量: | 516.37 |
| 类别: | Standards; Enzyme Activators and Inhibitors; |
| 应用: | XY 018 is a RORγ antagonist (EC50 = 190 nM). XY 018 suppresses androgen receptor expression in prostate cancer cell lines. Also inhibits growth of tumors in androgen receptor-positive xenograft models. |
| 参考文献 | |